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SIMM · NJU
Assay
PGDB_AS000640
System: biochemical
Target: BTRC | FBXW11 | SKP1
Assay context summary
Assay context
21 activity records
Assay family
biochemical
System
biochemical
Readout
EC50
Target
BTRC | FBXW11 | SKP1
E3
BTRC | FBXW11 | SKP1
Activity compounds and values
Activity records
21 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A009182
PGDB_C021142
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A015970
PGDB_C021135
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A019041
PGDB_C021139
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A019249
PGDB_C021148
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A023193
PGDB_C021138
PGDB_AS000640
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A024592
PGDB_C021147
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A025605
PGDB_C021143
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A030846
PGDB_C021140
PGDB_AS000640
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A032231
PGDB_C021146
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A033448
PGDB_C021149
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A056608
PGDB_C021137
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A058010
PGDB_C021144
PGDB_AS000640
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A060551
PGDB_C021140
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A063362
PGDB_C021134
PGDB_AS000640
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A065665
PGDB_C021133
PGDB_AS000640
View
EC50
-
<
1
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A068332
PGDB_C021146
PGDB_AS000640
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A069261
PGDB_C021141
PGDB_AS000640
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A071173
PGDB_C021133
PGDB_AS000640
View
EC50
-
=
1-10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A072828
PGDB_C021145
PGDB_AS000640
View
EC50
-
>
10
uM
-
—
CTNNB1
BTRC | FBXW11
-
WO2025179005A1
PGDB_A074878
PGDB_C021139
PGDB_AS000640
View