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Compound
PGDB_C029427
3 activity records1 related patents
2D structure
O=C1CCC(c2cccc(-c3ccc4c(c3)OCCCN4C(=O)c3ccccn3)c2Cl)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 84 | % | Concentration series: 10 uM, 1 uM | - | VAV1 | - | - | WO2026051943A1 | PGDB_A000135 | PGDB_C029427 | PGDB_AS000777 | View |
| DC50 | - | = | 8.4 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A000481 | PGDB_C029427 | PGDB_AS001440 | View |
| IC50 | - | = | 0.88 | nM | - | — | VAV1 | - | pan-T | WO2026051943A1 | PGDB_A002088 | PGDB_C029427 | PGDB_AS000112 | View |