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Compound
PGDB_C029452
3 activity records1 related patents
2D structure
Cn1cccc(N2CCCOc3cc(-c4cccc(C5CCC(=O)NC5=O)c4Cl)ccc32)c1=OCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 97.9 | % | Concentration series: 10 uM, 1 uM | - | VAV1 | - | - | WO2026051943A1 | PGDB_A000294 | PGDB_C029452 | PGDB_AS000777 | View |
| DC50 | - | = | 2.57 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A003116 | PGDB_C029452 | PGDB_AS001440 | View |
| IC50 | - | = | 0.13 | nM | - | — | VAV1 | - | pan-T | WO2026051943A1 | PGDB_A003681 | PGDB_C029452 | PGDB_AS000112 | View |