Assay
PGDB_AS000844
System: cell_basedCell line: NCI-H1975
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A015098 | PGDB_C025814 | PGDB_AS000844 | View | |
| IC50 | - | = | 50-100 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A016684 | PGDB_C025815 | PGDB_AS000844 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A034705 | PGDB_C025806 | PGDB_AS000844 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A036510 | PGDB_C025808 | PGDB_AS000844 | View | |
| IC50 | - | = | 50-100 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A046048 | PGDB_C025809 | PGDB_AS000844 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A056045 | PGDB_C025807 | PGDB_AS000844 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A071911 | PGDB_C019593 | PGDB_AS000844 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | NCI-H1975 | CN116239566A | PGDB_A072032 | PGDB_C015982 | PGDB_AS000844 | View |