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SIMM · NJU
Assay
PGDB_AS001067
System: cell_based
Target: GSPT1
Cell line: Jurkat
Assay context summary
Assay context
55 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
Target
GSPT1
E3
Not specified
Cell line
Jurkat
Technology
Western_blot
Activity compounds and values
Activity records
55 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A007081
PGDB_C001336
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A008236
PGDB_C001302
PGDB_AS001067
View
% Degradation
-
=
30-50
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A008778
PGDB_C001329
PGDB_AS001067
View
% Degradation
-
=
50-70
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A010634
PGDB_C001340
PGDB_AS001067
View
% Degradation
-
=
30-50
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A013421
PGDB_C001335
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A014279
PGDB_C001331
PGDB_AS001067
View
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A014348
PGDB_C001342
PGDB_AS001067
View
% Degradation
-
<=
30
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A014685
PGDB_C001357
PGDB_AS001067
View
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A015674
PGDB_C001303
PGDB_AS001067
View
% Degradation
-
=
30-50
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A016413
PGDB_C001352
PGDB_AS001067
View
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A018375
PGDB_C001332
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A018622
PGDB_C001326
PGDB_AS001067
View
% Degradation
-
<=
30
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A018846
PGDB_C001359
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A020517
PGDB_C001314
PGDB_AS001067
View
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A021841
PGDB_C001351
PGDB_AS001067
View
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A022107
PGDB_C001321
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A023658
PGDB_C001360
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A026795
PGDB_C001337
PGDB_AS001067
View
% Degradation
-
=
90-100
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A028526
PGDB_C001354
PGDB_AS001067
View
% Degradation
-
=
70-90
%
0.1 uM
24 h
GSPT1
-
Jurkat
WO2025110699A1
PGDB_A031440
PGDB_C001349
PGDB_AS001067
View