Assay context summary

Assay context

55 activity records
Activity compounds and values

Activity records

55 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C001336
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A007081PGDB_C001336PGDB_AS001067View
2D structure for PGDB_C001302
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A008236PGDB_C001302PGDB_AS001067View
2D structure for PGDB_C001329
% Degradation-=30-50%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A008778PGDB_C001329PGDB_AS001067View
2D structure for PGDB_C001340
% Degradation-=50-70%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A010634PGDB_C001340PGDB_AS001067View
2D structure for PGDB_C001335
% Degradation-=30-50%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A013421PGDB_C001335PGDB_AS001067View
2D structure for PGDB_C001331
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A014279PGDB_C001331PGDB_AS001067View
2D structure for PGDB_C001342
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A014348PGDB_C001342PGDB_AS001067View
2D structure for PGDB_C001357
% Degradation-<=30%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A014685PGDB_C001357PGDB_AS001067View
2D structure for PGDB_C001303
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A015674PGDB_C001303PGDB_AS001067View
2D structure for PGDB_C001352
% Degradation-=30-50%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A016413PGDB_C001352PGDB_AS001067View
2D structure for PGDB_C001332
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A018375PGDB_C001332PGDB_AS001067View
2D structure for PGDB_C001326
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A018622PGDB_C001326PGDB_AS001067View
2D structure for PGDB_C001359
% Degradation-<=30%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A018846PGDB_C001359PGDB_AS001067View
2D structure for PGDB_C001314
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A020517PGDB_C001314PGDB_AS001067View
2D structure for PGDB_C001351
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A021841PGDB_C001351PGDB_AS001067View
2D structure for PGDB_C001321
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A022107PGDB_C001321PGDB_AS001067View
2D structure for PGDB_C001360
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A023658PGDB_C001360PGDB_AS001067View
2D structure for PGDB_C001337
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A026795PGDB_C001337PGDB_AS001067View
2D structure for PGDB_C001354
% Degradation-=90-100%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A028526PGDB_C001354PGDB_AS001067View
2D structure for PGDB_C001349
% Degradation-=70-90%0.1 uM24 hGSPT1-JurkatWO2025110699A1PGDB_A031440PGDB_C001349PGDB_AS001067View