Assay context summary

Assay context

53 activity records
Activity compounds and values

Activity records

53 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019253
IC50-=1-5nM-IKZF3-MM.1RWO2025016359A1PGDB_A008554PGDB_C019253PGDB_AS001084View
2D structure for PGDB_C019222
IC50-=50-100nM-IKZF3-MM.1RWO2025016359A1PGDB_A010345PGDB_C019222PGDB_AS001084View
2D structure for PGDB_C019259
IC50-=1-5nM-IKZF3-MM.1RWO2025016359A1PGDB_A012623PGDB_C019259PGDB_AS001084View
2D structure for PGDB_C019186
IC50-=10-50nM-IKZF3-MM.1RWO2025016359A1PGDB_A012870PGDB_C019186PGDB_AS001084View
2D structure for PGDB_C019251
IC50-=1-5nM-IKZF3-MM.1RWO2025016359A1PGDB_A015602PGDB_C019251PGDB_AS001084View
2D structure for PGDB_C019252
IC50-=5-10nM-IKZF3-MM.1RWO2025016359A1PGDB_A016857PGDB_C019252PGDB_AS001084View
2D structure for PGDB_C019182
IC50-=5-10nM-IKZF3-MM.1RWO2025016359A1PGDB_A018374PGDB_C019182PGDB_AS001084View
2D structure for PGDB_C019235
IC50-=10-50nM-IKZF3-MM.1RWO2025016359A1PGDB_A020076PGDB_C019235PGDB_AS001084View
2D structure for PGDB_C019196
IC50-=10-50nM-IKZF3-MM.1RWO2025016359A1PGDB_A026042PGDB_C019196PGDB_AS001084View
2D structure for PGDB_C019250
IC50-=100-500nM-IKZF3-MM.1RWO2025016359A1PGDB_A026075PGDB_C019250PGDB_AS001084View
2D structure for PGDB_C019220
IC50-=10-50nM-IKZF3-MM.1RWO2025016359A1PGDB_A026189PGDB_C019220PGDB_AS001084View
2D structure for PGDB_C019227
IC50-=1-5nM-IKZF3-MM.1RWO2025016359A1PGDB_A026778PGDB_C019227PGDB_AS001084View
2D structure for PGDB_C019197
IC50-=10-50nM-IKZF3-MM.1RWO2025016359A1PGDB_A028619PGDB_C019197PGDB_AS001084View
2D structure for PGDB_C019221
IC50-=1-5nM-IKZF3-MM.1RWO2025016359A1PGDB_A028702PGDB_C019221PGDB_AS001084View
2D structure for PGDB_C019256
IC50-<1nM-IKZF3-MM.1RWO2025016359A1PGDB_A028832PGDB_C019256PGDB_AS001084View
2D structure for PGDB_C019195
IC50-=5-10nM-IKZF3-MM.1RWO2025016359A1PGDB_A031259PGDB_C019195PGDB_AS001084View
2D structure for PGDB_C019236
IC50-=10-50nM-IKZF3-MM.1RWO2025016359A1PGDB_A031569PGDB_C019236PGDB_AS001084View
2D structure for PGDB_C019181
IC50-=5-10nM-IKZF3-MM.1RWO2025016359A1PGDB_A031872PGDB_C019181PGDB_AS001084View
2D structure for PGDB_C019232
IC50-=50-100nM-IKZF3-MM.1RWO2025016359A1PGDB_A032278PGDB_C019232PGDB_AS001084View
2D structure for PGDB_C019200
IC50-=1-5nM-IKZF3-MM.1RWO2025016359A1PGDB_A032350PGDB_C019200PGDB_AS001084View