Assay
PGDB_AS001097
System: cell_basedTarget: IKZF3Cell line: NCI-H929
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 77.1 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A009731 | PGDB_C025617 | PGDB_AS001097 | View | |
| Dmax | - | = | 71.4 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A010422 | PGDB_C025597 | PGDB_AS001097 | View | |
| Dmax | - | = | 76.4 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A010531 | PGDB_C025616 | PGDB_AS001097 | View | |
| Dmax | - | = | 76.2 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A027390 | PGDB_C025619 | PGDB_AS001097 | View | |
| Dmax | - | = | 76.6 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A028222 | PGDB_C025599 | PGDB_AS001097 | View | |
| Dmax | - | = | 75 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A038635 | PGDB_C021276 | PGDB_AS001097 | View | |
| Dmax | - | = | 70.3 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A045080 | PGDB_C025600 | PGDB_AS001097 | View | |
| Dmax | - | = | 74.1 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A058978 | PGDB_C025615 | PGDB_AS001097 | View | |
| Dmax | - | = | 73.8 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A060010 | PGDB_C025601 | PGDB_AS001097 | View | |
| Dmax | - | = | 73.2 | % | Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM | 24 h | IKZF3 | - | NCI-H929 | CA3286762A1 | PGDB_A070777 | PGDB_C021277 | PGDB_AS001097 | View |