Assay context summary

Assay context

10 activity records
Activity compounds and values

Activity records

10 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C025617
Dmax-=77.1%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A009731PGDB_C025617PGDB_AS001097View
2D structure for PGDB_C025597
Dmax-=71.4%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A010422PGDB_C025597PGDB_AS001097View
2D structure for PGDB_C025616
Dmax-=76.4%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A010531PGDB_C025616PGDB_AS001097View
2D structure for PGDB_C025619
Dmax-=76.2%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A027390PGDB_C025619PGDB_AS001097View
2D structure for PGDB_C025599
Dmax-=76.6%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A028222PGDB_C025599PGDB_AS001097View
2D structure for PGDB_C021276
Dmax-=75%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A038635PGDB_C021276PGDB_AS001097View
2D structure for PGDB_C025600
Dmax-=70.3%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A045080PGDB_C025600PGDB_AS001097View
2D structure for PGDB_C025615
Dmax-=74.1%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A058978PGDB_C025615PGDB_AS001097View
2D structure for PGDB_C025601
Dmax-=73.8%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A060010PGDB_C025601PGDB_AS001097View
2D structure for PGDB_C021277
Dmax-=73.2%Concentration series: 1600 nM, 400 nM, 100 nM, 25 nM, 6.25 nM, 1.56 nM, 0.39 nM, 0.1 nM24 hIKZF3-NCI-H929CA3286762A1PGDB_A070777PGDB_C021277PGDB_AS001097View