Assay

PGDB_AS001130

System: biochemicalTarget: CRBN | DDB1
Assay context summary

Assay context

28 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetCRBN | DDB1
E3CRBN | DDB1
TechnologyHTRF
Activity compounds and values

Activity records

28 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C009038
IC50-=1-10uM-—CRBNCRBN-US12540127B2PGDB_A012655PGDB_C009038PGDB_AS001130View
2D structure for PGDB_C009034
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A013802PGDB_C009034PGDB_AS001130View
2D structure for PGDB_C009047
IC50-=1-10uM-—CRBNCRBN-US12540127B2PGDB_A015418PGDB_C009047PGDB_AS001130View
2D structure for PGDB_C009035
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A024195PGDB_C009035PGDB_AS001130View
2D structure for PGDB_C009039
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A024343PGDB_C009039PGDB_AS001130View
2D structure for PGDB_C009051
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A027283PGDB_C009051PGDB_AS001130View
2D structure for PGDB_C009036
IC50-=10-100uM-—CRBNCRBN-US12540127B2PGDB_A028686PGDB_C009036PGDB_AS001130View
2D structure for PGDB_C009057
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A031399PGDB_C009057PGDB_AS001130View
2D structure for PGDB_C009046
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A038440PGDB_C009046PGDB_AS001130View
2D structure for PGDB_C009040
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A041299PGDB_C009040PGDB_AS001130View
2D structure for PGDB_C009048
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A043509PGDB_C009048PGDB_AS001130View
2D structure for PGDB_C009050
IC50-=10-100uM-—CRBNCRBN-US12540127B2PGDB_A046935PGDB_C009050PGDB_AS001130View
2D structure for PGDB_C009061
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A047564PGDB_C009061PGDB_AS001130View
2D structure for PGDB_C009058
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A048235PGDB_C009058PGDB_AS001130View
2D structure for PGDB_C009042
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A048466PGDB_C009042PGDB_AS001130View
2D structure for PGDB_C009041
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A050333PGDB_C009041PGDB_AS001130View
2D structure for PGDB_C009044
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A053077PGDB_C009044PGDB_AS001130View
2D structure for PGDB_C009052
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A053431PGDB_C009052PGDB_AS001130View
2D structure for PGDB_C009037
IC50-=1-10uM-—CRBNCRBN-US12540127B2PGDB_A053524PGDB_C009037PGDB_AS001130View
2D structure for PGDB_C009049
IC50-<1uM-—CRBNCRBN-US12540127B2PGDB_A057493PGDB_C009049PGDB_AS001130View
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