Assay
PGDB_AS001148
System: cell_basedCell line: MM.1S
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A027517 | PGDB_C025822 | PGDB_AS001148 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A042040 | PGDB_C019594 | PGDB_AS001148 | View | |
| IC50 | - | > | 10000 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A050945 | PGDB_C025816 | PGDB_AS001148 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | MM.1S | CN116239566A | PGDB_A068824 | PGDB_C025818 | PGDB_AS001148 | View |