Assay

PGDB_AS001173

System: cell_basedTarget: GSPT1Cell line: HL-60
Assay context summary

Assay context

28 activity records
Assay family% Degradation
Systemcell_based
Readout% Degradation
TargetGSPT1
E3Not specified
Cell lineHL-60
TechnologyWestern_blot
Detection targetprotein_degradation
Activity compounds and values

Activity records

28 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C002853
% Degradation-=0%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A020268PGDB_C002853PGDB_AS001173View
2D structure for PGDB_C002877
% Degradation-=95%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A022297PGDB_C002877PGDB_AS001173View
2D structure for PGDB_C002851
% Degradation-=0%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A022945PGDB_C002851PGDB_AS001173View
2D structure for PGDB_C002857
% Degradation-=63%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A023659PGDB_C002857PGDB_AS001173View
2D structure for PGDB_C002871
% Degradation-=29%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A023672PGDB_C002871PGDB_AS001173View
2D structure for PGDB_C002865
% Degradation-=32%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A023676PGDB_C002865PGDB_AS001173View
2D structure for PGDB_C002870
% Degradation-=40%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A023810PGDB_C002870PGDB_AS001173View
2D structure for PGDB_C002855
% Degradation-=52%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A024451PGDB_C002855PGDB_AS001173View
2D structure for PGDB_C002876
% Degradation-=90%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A027064PGDB_C002876PGDB_AS001173View
2D structure for PGDB_C002858
% Degradation-=15%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A031542PGDB_C002858PGDB_AS001173View
2D structure for PGDB_C002868
% Degradation-=38%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A032392PGDB_C002868PGDB_AS001173View
2D structure for PGDB_C002874
% Degradation->95%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A037253PGDB_C002874PGDB_AS001173View
2D structure for PGDB_C002875
% Degradation-=75%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A043078PGDB_C002875PGDB_AS001173View
2D structure for PGDB_C002850
% Degradation-=51%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A046781PGDB_C002850PGDB_AS001173View
2D structure for PGDB_C002859
% Degradation-=45%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A047281PGDB_C002859PGDB_AS001173View
2D structure for PGDB_C002866
% Degradation-=22%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A047922PGDB_C002866PGDB_AS001173View
2D structure for PGDB_C002864
% Degradation-=57%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A056960PGDB_C002864PGDB_AS001173View
2D structure for PGDB_C002867
% Degradation-=36%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A057295PGDB_C002867PGDB_AS001173View
2D structure for PGDB_C002860
% Degradation-<5%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A057980PGDB_C002860PGDB_AS001173View
2D structure for PGDB_C002856
% Degradation-=10%1 uM2 hGSPT1-HL-60WO2024073871A1PGDB_A062153PGDB_C002856PGDB_AS001173View
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