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Compound
PGDB_C002875
3 activity records1 related patents
2D structure
O=C1CCC(N2C(=O)c3cc(F)c(N4CCC(CCN5CCCN(c6cccc(-c7cnc8[nH]cc(C9CC9)c8c7Cl)c6)C5=O)CC4)cc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 122 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A035575 | PGDB_C002875 | PGDB_AS000219 | View |
| % Degradation | - | = | 45 | % | 0.1 uM | 2 h | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A042909 | PGDB_C002875 | PGDB_AS000569 | View |
| % Degradation | - | = | 75 | % | 1 uM | 2 h | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A043078 | PGDB_C002875 | PGDB_AS001173 | View |