Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C002876
3 activity records1 related patents
2D structure
CCc1c[nH]c2ncc(-c3cccc(N4CCCN(CCNc5ccc6c(c5)C(=O)N(C5CCC(=O)NC5=O)C6=O)C4=O)c3)c(Cl)c12Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 23 | nM | - | — | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A017879 | PGDB_C002876 | PGDB_AS000219 | View |
| % Degradation | - | = | 90 | % | 1 uM | 2 h | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A027064 | PGDB_C002876 | PGDB_AS001173 | View |
| % Degradation | - | = | 63 | % | 0.1 uM | 2 h | GSPT1 | - | HL-60 | WO2024073871A1 | PGDB_A057329 | PGDB_C002876 | PGDB_AS000569 | View |