Assay
PGDB_AS001192
System: cell_basedCell line: SW620
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 717 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A036163 | PGDB_C001179 | PGDB_AS001192 | View | |
| IC50 | - | = | 708.8 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A038331 | PGDB_C001180 | PGDB_AS001192 | View | |
| IC50 | - | = | 18.6 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A041851 | PGDB_C001156 | PGDB_AS001192 | View | |
| IC50 | - | > | 10000 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A067776 | PGDB_C008731 | PGDB_AS001192 | View | |
| IC50 | - | = | 35.8 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A068746 | PGDB_C001158 | PGDB_AS001192 | View | |
| IC50 | - | = | 386.8 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A074395 | PGDB_C001178 | PGDB_AS001192 | View |