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Cc1nc2cccc(SCCCN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)c2c(=O)n1C1CCC(=O)NC1=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 12.7 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A009697 | PGDB_C001156 | PGDB_AS001111 | View | |
| IC50 | - | = | 44.9 | nM | - | — | - | - | Daudi | WO2023151635A1 | PGDB_A011353 | PGDB_C001156 | PGDB_AS000279 | View | |
| IC50 | - | = | 86.5 | nM | - | — | - | - | TMD8 | WO2023151635A1 | PGDB_A013204 | PGDB_C001156 | PGDB_AS000648 | View | |
| IC50 | - | = | 29.3 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A027216 | PGDB_C001156 | PGDB_AS002383 | View | |
| IC50 | - | = | 18.6 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A041851 | PGDB_C001156 | PGDB_AS001192 | View | |
| IC50 | - | = | 22.3 | nM | - | — | - | - | Kasumi-1 | WO2023151635A1 | PGDB_A042294 | PGDB_C001156 | PGDB_AS001646 | View | |
| IC50 | - | = | 89.3 | nM | - | — | - | - | Ramos | WO2023151635A1 | PGDB_A057455 | PGDB_C001156 | PGDB_AS002135 | View | |
| IC50 | - | = | 1.57 | uM | - | — | CRBN | CRBN | - | WO2023151635A1 | PGDB_A075905 | PGDB_C001156 | PGDB_AS000788 | View |