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Cc1nc2ccc(NCCN3CCN(CCC45CC6CC(CC(C6)C4)C5)CC3)cc2c(=O)n1C1CCC(=O)NC1=O| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 1.72 | uM | - | — | CRBN | CRBN | - | WO2023151635A1 | PGDB_A009503 | PGDB_C001158 | PGDB_AS000788 | View | |
| IC50 | - | = | 32.8 | nM | - | — | - | - | MM.1R | WO2023151635A1 | PGDB_A015334 | PGDB_C001158 | PGDB_AS001111 | View | |
| IC50 | - | = | 164.7 | nM | - | — | - | - | Ramos | WO2023151635A1 | PGDB_A018178 | PGDB_C001158 | PGDB_AS002135 | View | |
| IC50 | - | = | 79.6 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A025202 | PGDB_C001158 | PGDB_AS002383 | View | |
| IC50 | - | = | 155.4 | nM | - | — | - | - | Daudi | WO2023151635A1 | PGDB_A043448 | PGDB_C001158 | PGDB_AS000279 | View | |
| IC50 | - | = | 185.8 | nM | - | — | - | - | TMD8 | WO2023151635A1 | PGDB_A066021 | PGDB_C001158 | PGDB_AS000648 | View | |
| IC50 | - | = | 35.8 | nM | - | — | - | - | SW620 | WO2023151635A1 | PGDB_A068746 | PGDB_C001158 | PGDB_AS001192 | View | |
| IC50 | - | = | 104.1 | nM | - | — | - | - | Kasumi-1 | WO2023151635A1 | PGDB_A071429 | PGDB_C001158 | PGDB_AS001646 | View |