Assay
PGDB_AS001230
System: cell_basedCell line: Kasumi-1
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A012076 | PGDB_C025962 | PGDB_AS001230 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A021420 | PGDB_C019639 | PGDB_AS001230 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A039971 | PGDB_C025964 | PGDB_AS001230 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A049498 | PGDB_C025954 | PGDB_AS001230 | View | |
| IC50 | - | = | 50-100 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A049988 | PGDB_C025963 | PGDB_AS001230 | View | |
| IC50 | - | = | 50-100 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A050637 | PGDB_C025966 | PGDB_AS001230 | View | |
| IC50 | - | = | 100-500 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A055468 | PGDB_C025961 | PGDB_AS001230 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A055979 | PGDB_C025953 | PGDB_AS001230 | View | |
| IC50 | - | < | 50 | nM | - | — | IRAK4 | - | Kasumi-1 | CN116239566A | PGDB_A065909 | PGDB_C025965 | PGDB_AS001230 | View |