Assay
PGDB_AS001305
System: cell_basedCell line: SW620
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A007820 | PGDB_C019594 | PGDB_AS001305 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A016074 | PGDB_C019596 | PGDB_AS001305 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A017356 | PGDB_C025818 | PGDB_AS001305 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A031759 | PGDB_C025823 | PGDB_AS001305 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A045847 | PGDB_C025822 | PGDB_AS001305 | View | |
| IC50 | - | < | 50 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A047790 | PGDB_C025824 | PGDB_AS001305 | View | |
| IC50 | - | = | 100-500 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A068992 | PGDB_C019597 | PGDB_AS001305 | View | |
| IC50 | - | = | 50-100 | nM | - | — | ESR1 | - | SW620 | CN116239566A | PGDB_A069916 | PGDB_C025826 | PGDB_AS001305 | View |