Assay context summary

Assay context

15 activity records
Activity compounds and values

Activity records

15 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C005465
IC50-=20.27nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A007288PGDB_C005465PGDB_AS001340View
2D structure for PGDB_C005468
IC50-=22.92nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A010357PGDB_C005468PGDB_AS001340View
2D structure for PGDB_C005462
IC50-=78.93nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A011256PGDB_C005462PGDB_AS001340View
2D structure for PGDB_C005472
IC50-=25.94nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A012477PGDB_C005472PGDB_AS001340View
2D structure for PGDB_C005469
IC50-=98.66nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A022285PGDB_C005469PGDB_AS001340View
2D structure for PGDB_C003382
IC50-=121.46nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A024823PGDB_C003382PGDB_AS001340View
2D structure for PGDB_C005473
IC50-=26.62nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A035788PGDB_C005473PGDB_AS001340View
2D structure for PGDB_C005475
IC50-=194.82nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A036698PGDB_C005475PGDB_AS001340View
2D structure for PGDB_C005466
IC50-=5.182nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A039030PGDB_C005466PGDB_AS001340View
2D structure for PGDB_C005467
IC50-=5.39nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A052282PGDB_C005467PGDB_AS001340View
2D structure for PGDB_C005474
IC50-=23.23nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A059410PGDB_C005474PGDB_AS001340View
2D structure for PGDB_C005463
IC50-=220.1nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A066842PGDB_C005463PGDB_AS001340View
2D structure for PGDB_C005470
IC50-=6.77nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A069146PGDB_C005470PGDB_AS001340View
2D structure for PGDB_C005471
IC50-=3.88nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A074361PGDB_C005471PGDB_AS001340View
2D structure for PGDB_C005464
IC50-=7.586nM-GSPT1-SK-BR-3WO2025252247A1PGDB_A076871PGDB_C005464PGDB_AS001340View