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Compound
PGDB_C029470
4 activity records2 related patents
2D structure
Cn1ccc(CN2C(=O)C3(CC3)Oc3cc(-c4cccc(C5CCC(=O)NC5=O)c4Cl)ccc32)n1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 3.46 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A000558 | PGDB_C029470 | PGDB_AS001440 | View |
| DC50 | - | = | 31.86 | nM | - | — | VAV1 | - | 293T-VAV1-FLAG | WO2026103873A1 | PGDB_A000709 | PGDB_C029470 | PGDB_AS000831 | View |
| IC50 | - | = | 0.06 | nM | - | — | VAV1 | - | pan-T | WO2026051943A1 | PGDB_A002797 | PGDB_C029470 | PGDB_AS000112 | View |
| Dmax | - | = | 98.11 | % | Concentration series: 10 uM, 1 uM | - | VAV1 | - | - | WO2026051943A1 | PGDB_A081255 | PGDB_C029470 | PGDB_AS000777 | View |