Assay context summary

Assay context

31 activity records
Activity compounds and values

Activity records

31 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C019201
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A009387PGDB_C019201PGDB_AS001811View
2D structure for PGDB_C019193
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A009477PGDB_C019193PGDB_AS001811View
2D structure for PGDB_C019181
IC50-=50-100nM-IKZF3-SW620WO2025016359A1PGDB_A010342PGDB_C019181PGDB_AS001811View
2D structure for PGDB_C019198
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A013274PGDB_C019198PGDB_AS001811View
2D structure for PGDB_C019199
IC50-=10-50nM-IKZF3-SW620WO2025016359A1PGDB_A014840PGDB_C019199PGDB_AS001811View
2D structure for PGDB_C019200
IC50-=10-50nM-IKZF3-SW620WO2025016359A1PGDB_A017659PGDB_C019200PGDB_AS001811View
2D structure for PGDB_C019222
IC50-=500-1000nM-IKZF3-SW620WO2025016359A1PGDB_A019256PGDB_C019222PGDB_AS001811View
2D structure for PGDB_C019191
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A021857PGDB_C019191PGDB_AS001811View
2D structure for PGDB_C019212
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A026272PGDB_C019212PGDB_AS001811View
2D structure for PGDB_C019195
IC50-=10-50nM-IKZF3-SW620WO2025016359A1PGDB_A031414PGDB_C019195PGDB_AS001811View
2D structure for PGDB_C019220
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A032225PGDB_C019220PGDB_AS001811View
2D structure for PGDB_C019186
IC50-=500-1000nM-IKZF3-SW620WO2025016359A1PGDB_A033361PGDB_C019186PGDB_AS001811View
2D structure for PGDB_C019175
IC50-=50-100nM-IKZF3-SW620WO2025016359A1PGDB_A033905PGDB_C019175PGDB_AS001811View
2D structure for PGDB_C019196
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A035770PGDB_C019196PGDB_AS001811View
2D structure for PGDB_C019190
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A036062PGDB_C019190PGDB_AS001811View
2D structure for PGDB_C019204
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A036714PGDB_C019204PGDB_AS001811View
2D structure for PGDB_C019194
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A037123PGDB_C019194PGDB_AS001811View
2D structure for PGDB_C019182
IC50-=50-100nM-IKZF3-SW620WO2025016359A1PGDB_A037205PGDB_C019182PGDB_AS001811View
2D structure for PGDB_C019228
IC50-=100-500nM-IKZF3-SW620WO2025016359A1PGDB_A038748PGDB_C019228PGDB_AS001811View
2D structure for PGDB_C019218
IC50-=5-10nM-IKZF3-SW620WO2025016359A1PGDB_A039990PGDB_C019218PGDB_AS001811View