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SIMM · NJU
Assay
PGDB_AS001956
System: cell_based
Target: NEK7
Assay context summary
Assay context
19 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
Target
NEK7
E3
CRBN
Activity compounds and values
Activity records
19 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
60
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A010068
PGDB_C020453
PGDB_AS001956
View
Dmax
-
=
79
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A019569
PGDB_C020449
PGDB_AS001956
View
Dmax
-
=
82
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A023172
PGDB_C020439
PGDB_AS001956
View
Dmax
-
=
61
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A023610
PGDB_C020448
PGDB_AS001956
View
Dmax
-
=
3
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A025820
PGDB_C020447
PGDB_AS001956
View
Dmax
-
=
70
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A026780
PGDB_C020446
PGDB_AS001956
View
Dmax
-
=
88
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A034248
PGDB_C020438
PGDB_AS001956
View
Dmax
-
=
68
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A040974
PGDB_C020444
PGDB_AS001956
View
Dmax
-
=
94
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A046676
PGDB_C020440
PGDB_AS001956
View
Dmax
-
=
78
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A057810
PGDB_C020455
PGDB_AS001956
View
Dmax
-
=
67
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A058180
PGDB_C020454
PGDB_AS001956
View
Dmax
-
=
68
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A058589
PGDB_C020437
PGDB_AS001956
View
Dmax
-
=
90
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A059367
PGDB_C020436
PGDB_AS001956
View
Dmax
-
=
71
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A063564
PGDB_C020451
PGDB_AS001956
View
Dmax
-
=
88
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A063638
PGDB_C020435
PGDB_AS001956
View
Dmax
-
=
95
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A064011
PGDB_C020442
PGDB_AS001956
View
Dmax
-
=
61
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A065143
PGDB_C020450
PGDB_AS001956
View
Dmax
-
=
57
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A074095
PGDB_C020445
PGDB_AS001956
View
Dmax
-
=
54
%
-
-
NEK7
CRBN
-
WO2025024521A1
PGDB_A076754
PGDB_C020452
PGDB_AS001956
View