Assay
PGDB_AS001968
System: cell_basedTarget: CRBNCell line: NCI-H1155
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 25 | nM | - | — | CRBN | CRBN | NCI-H1155 | WO2024125437A1 | PGDB_A018808 | PGDB_C001479 | PGDB_AS001968 | View | |
| IC50 | - | = | 57 | nM | - | — | CRBN | CRBN | NCI-H1155 | WO2024125437A1 | PGDB_A027361 | PGDB_C000378 | PGDB_AS001968 | View | |
| IC50 | - | = | 141 | nM | - | — | CRBN | CRBN | NCI-H1155 | WO2024125437A1 | PGDB_A033648 | PGDB_C021942 | PGDB_AS001968 | View | |
| IC50 | - | = | 31.1 | nM | - | — | CRBN | CRBN | NCI-H1155 | WO2024125437A1 | PGDB_A038008 | PGDB_C005371 | PGDB_AS001968 | View |