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SIMM · NJU
Assay
PGDB_AS002054
System: biochemical
Target: RAF1 | SOS1
Assay context summary
Assay context
41 activity records
Assay family
biochemical
System
biochemical
Readout
IC50
Target
RAF1 | SOS1
E3
Not specified
Technology
HTRF
Activity compounds and values
Activity records
41 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A007755
PGDB_C011617
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A008365
PGDB_C011625
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A009797
PGDB_C011624
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A011953
PGDB_C011597
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A013478
PGDB_C011628
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A014023
PGDB_C011615
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A014253
PGDB_C011595
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A015997
PGDB_C011588
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A016355
PGDB_C011624
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A018521
PGDB_C011593
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A019578
PGDB_C011630
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A019618
PGDB_C011596
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A020979
PGDB_C011606
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A022097
PGDB_C011607
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A023570
PGDB_C011591
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A023669
PGDB_C011605
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A024887
PGDB_C011616
PGDB_AS002054
View
IC50
-
=
10-100
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A026904
PGDB_C011620
PGDB_AS002054
View
IC50
-
=
100-1000
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A027575
PGDB_C011622
PGDB_AS002054
View
IC50
-
=
1-10
nM
-
—
KRAS
-
-
WO2025214350A1
PGDB_A027600
PGDB_C011627
PGDB_AS002054
View