Assay context summary

Assay context

41 activity records
Activity compounds and values

Activity records

41 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C011617
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A007755PGDB_C011617PGDB_AS002054View
2D structure for PGDB_C011625
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A008365PGDB_C011625PGDB_AS002054View
2D structure for PGDB_C011624
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A009797PGDB_C011624PGDB_AS002054View
2D structure for PGDB_C011597
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A011953PGDB_C011597PGDB_AS002054View
2D structure for PGDB_C011628
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A013478PGDB_C011628PGDB_AS002054View
2D structure for PGDB_C011615
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A014023PGDB_C011615PGDB_AS002054View
2D structure for PGDB_C011595
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A014253PGDB_C011595PGDB_AS002054View
2D structure for PGDB_C011588
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A015997PGDB_C011588PGDB_AS002054View
2D structure for PGDB_C011624
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A016355PGDB_C011624PGDB_AS002054View
2D structure for PGDB_C011593
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A018521PGDB_C011593PGDB_AS002054View
2D structure for PGDB_C011630
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A019578PGDB_C011630PGDB_AS002054View
2D structure for PGDB_C011596
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A019618PGDB_C011596PGDB_AS002054View
2D structure for PGDB_C011606
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A020979PGDB_C011606PGDB_AS002054View
2D structure for PGDB_C011607
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A022097PGDB_C011607PGDB_AS002054View
2D structure for PGDB_C011591
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A023570PGDB_C011591PGDB_AS002054View
2D structure for PGDB_C011605
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A023669PGDB_C011605PGDB_AS002054View
2D structure for PGDB_C011616
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A024887PGDB_C011616PGDB_AS002054View
2D structure for PGDB_C011620
IC50-=10-100nM-KRAS--WO2025214350A1PGDB_A026904PGDB_C011620PGDB_AS002054View
2D structure for PGDB_C011622
IC50-=100-1000nM-KRAS--WO2025214350A1PGDB_A027575PGDB_C011622PGDB_AS002054View
2D structure for PGDB_C011627
IC50-=1-10nM-KRAS--WO2025214350A1PGDB_A027600PGDB_C011627PGDB_AS002054View