Assay

PGDB_AS002060

System: biochemicalTarget: CDK12
Assay context summary

Assay context

12 activity records
Assay familybiochemical
Systembiochemical
ReadoutIC50
TargetCDK12
E3Not specified
Activity compounds and values

Activity records

12 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C007326
IC50-=19.37nM-—CDK12--CN121108130APGDB_A008223PGDB_C007326PGDB_AS002060View
2D structure for PGDB_C007335
IC50-=57.46nM-—CDK12--CN121108130APGDB_A008550PGDB_C007335PGDB_AS002060View
2D structure for PGDB_C007328
IC50-=31.52nM-—CDK12--CN121108130APGDB_A010946PGDB_C007328PGDB_AS002060View
2D structure for PGDB_C007333
IC50->10000nM-—CDK12--CN121108130APGDB_A022810PGDB_C007333PGDB_AS002060View
2D structure for PGDB_C007325
IC50-=34.54nM-—CDK12--CN121108130APGDB_A028513PGDB_C007325PGDB_AS002060View
2D structure for PGDB_C007331
IC50-=17.51nM-—CDK12--CN121108130APGDB_A031523PGDB_C007331PGDB_AS002060View
2D structure for PGDB_C007334
IC50-=34.21nM-—CDK12--CN121108130APGDB_A055380PGDB_C007334PGDB_AS002060View
2D structure for PGDB_C007330
IC50-=50.66nM-—CDK12--CN121108130APGDB_A056721PGDB_C007330PGDB_AS002060View
2D structure for PGDB_C007164
IC50-=101.28nM-—CDK12--CN121108130APGDB_A062326PGDB_C007164PGDB_AS002060View
2D structure for PGDB_C007329
IC50-=107.68nM-—CDK12--CN121108130APGDB_A070978PGDB_C007329PGDB_AS002060View
2D structure for PGDB_C007332
IC50-=118.93nM-—CDK12--CN121108130APGDB_A073041PGDB_C007332PGDB_AS002060View
2D structure for PGDB_C007327
IC50->10000nM-—CDK12--CN121108130APGDB_A073890PGDB_C007327PGDB_AS002060View
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