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C=CC(=O)Nc1ccccc1-c1ccc2nc(CC(=O)Nc3cc(C4CC4)[nH]n3)cn2n1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 351.6 | nM | - | — | CDK12 | - | MDA-MB-231 | CN121108130A | PGDB_A031323 | PGDB_C007329 | PGDB_AS001069 | View | |
| IC50 | - | = | 504.2 | nM | - | — | CDK12 | - | MDA-MB-468 | CN121108130A | PGDB_A069910 | PGDB_C007329 | PGDB_AS000556 | View | |
| IC50 | - | = | 107.68 | nM | - | — | CDK12 | - | - | CN121108130A | PGDB_A070978 | PGDB_C007329 | PGDB_AS002060 | View |