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C=CC(=O)Nc1ccc(-c2ccc3nc(CC(=O)Nc4ncc(C(C)(C)C)s4)cn3n2)cc1F| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 57.46 | nM | - | — | CDK12 | - | - | CN121108130A | PGDB_A008550 | PGDB_C007335 | PGDB_AS002060 | View | |
| IC50 | - | = | 219 | nM | - | — | CDK12 | - | MDA-MB-231 | CN121108130A | PGDB_A033466 | PGDB_C007335 | PGDB_AS001069 | View | |
| IC50 | - | = | 353.7 | nM | - | — | CDK12 | - | MDA-MB-468 | CN121108130A | PGDB_A044111 | PGDB_C007335 | PGDB_AS000556 | View |