Assay

PGDB_AS002100

System: cell_basedTarget: CDK2Cell line: HEK293
Assay context summary

Assay context

94 activity records
Assay family% Degradation
Systemcell_based
ReadoutIC50
TargetCDK2
E3Not specified
Cell lineHEK293
OrganismHomo sapiens
Technologyluminescence
Detection targetprotein_degradation
Activity compounds and values

Activity records

94 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008081
IC50-=0.0078uM-—CDK2-HEK293WO2025043225PGDB_A009011PGDB_C008081PGDB_AS002100View
2D structure for PGDB_C008071
IC50-=0.057uM-—CDK2-HEK293WO2025043225PGDB_A009404PGDB_C008071PGDB_AS002100View
2D structure for PGDB_C008135
IC50-=0.02uM-—CDK2-HEK293WO2025043225PGDB_A013293PGDB_C008135PGDB_AS002100View
2D structure for PGDB_C008120
IC50-=0.0065uM-—CDK2-HEK293WO2025043225PGDB_A016042PGDB_C008120PGDB_AS002100View
2D structure for PGDB_C008106
IC50-=0.11uM-—CDK2-HEK293WO2025043225PGDB_A016594PGDB_C008106PGDB_AS002100View
2D structure for PGDB_C008066
IC50-=0.031uM-—CDK2-HEK293WO2025043225PGDB_A017048PGDB_C008066PGDB_AS002100View
2D structure for PGDB_C008117
IC50-=0.0048uM-—CDK2-HEK293WO2025043225PGDB_A017492PGDB_C008117PGDB_AS002100View
2D structure for PGDB_C008051
IC50-=0.031uM-—CDK2-HEK293WO2025043225PGDB_A017734PGDB_C008051PGDB_AS002100View
2D structure for PGDB_C008087
IC50-=0.07uM-—CDK2-HEK293WO2025043225PGDB_A018045PGDB_C008087PGDB_AS002100View
2D structure for PGDB_C008088
IC50-=0.025uM-—CDK2-HEK293WO2025043225PGDB_A018344PGDB_C008088PGDB_AS002100View
2D structure for PGDB_C008047
IC50-=0.041uM-—CDK2-HEK293WO2025043225PGDB_A018543PGDB_C008047PGDB_AS002100View
2D structure for PGDB_C008095
IC50-=0.021uM-—CDK2-HEK293WO2025043225PGDB_A018643PGDB_C008095PGDB_AS002100View
2D structure for PGDB_C008090
IC50-=0.098uM-—CDK2-HEK293WO2025043225PGDB_A018818PGDB_C008090PGDB_AS002100View
2D structure for PGDB_C008054
IC50-=0.0095uM-—CDK2-HEK293WO2025043225PGDB_A019133PGDB_C008054PGDB_AS002100View
2D structure for PGDB_C008076
IC50-=0.034uM-—CDK2-HEK293WO2025043225PGDB_A019276PGDB_C008076PGDB_AS002100View
2D structure for PGDB_C008125
IC50-=0.12uM-—CDK2-HEK293WO2025043225PGDB_A019787PGDB_C008125PGDB_AS002100View
2D structure for PGDB_C008137
IC50-=0.041uM-—CDK2-HEK293WO2025043225PGDB_A020005PGDB_C008137PGDB_AS002100View
2D structure for PGDB_C008097
IC50-=0.0029uM-—CDK2-HEK293WO2025043225PGDB_A020568PGDB_C008097PGDB_AS002100View
2D structure for PGDB_C008079
IC50-=0.035uM-—CDK2-HEK293WO2025043225PGDB_A022823PGDB_C008079PGDB_AS002100View
2D structure for PGDB_C008049
IC50-=0.053uM-—CDK2-HEK293WO2025043225PGDB_A024762PGDB_C008049PGDB_AS002100View
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