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SIMM · NJU
Assay
PGDB_AS002152
System: biochemical
Target: CRBN | DDB1
Assay context summary
Assay context
113 activity records
Assay family
ternary_complex
System
biochemical
Readout
Fold change
Target
CRBN | DDB1
E3
CRBN | DDB1
Activity compounds and values
Activity records
113 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
=
100-1000
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A007242
PGDB_C012275
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A007728
PGDB_C012380
PGDB_AS002152
View
EC50
-
<
10
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A008993
PGDB_C012320
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A009912
PGDB_C012388
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A010507
PGDB_C012280
PGDB_AS002152
View
EC50
-
=
100-1000
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A010670
PGDB_C012316
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A012366
PGDB_C012323
PGDB_AS002152
View
EC50
-
=
100-1000
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A012805
PGDB_C012276
PGDB_AS002152
View
EC50
-
>
1000
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A012930
PGDB_C012340
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A013110
PGDB_C012381
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A013153
PGDB_C012274
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A014532
PGDB_C012385
PGDB_AS002152
View
EC50
-
>
1000
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A015008
PGDB_C012366
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A015172
PGDB_C012398
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A015877
PGDB_C012401
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A016486
PGDB_C012329
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A016525
PGDB_C012327
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A018765
PGDB_C012322
PGDB_AS002152
View
EC50
-
=
100-1000
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A019576
PGDB_C012278
PGDB_AS002152
View
EC50
-
=
10-100
nM
-
—
ALK
CRBN
-
WO2026015344A1
PGDB_A019838
PGDB_C012386
PGDB_AS002152
View