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NCc1ccc(-c2noc(CN3CCCC4=C3C(=O)N(C3CCC(=O)NC3=O)C4=O)n2)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | > | 1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A012930 | PGDB_C012340 | PGDB_AS002152 | View | |
| EC50 | - | > | 1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A028974 | PGDB_C012340 | PGDB_AS000738 | View | |
| Emax | - | < | 50 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A048783 | PGDB_C012340 | PGDB_AS001094 | View | |
| Emax | - | < | 50 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A074214 | PGDB_C012340 | PGDB_AS001769 | View |