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O=C1CCC(N2C(=O)C3=C(C2=O)N(Cc2ccc4ccccc4c2)CCC3)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| EC50 | - | = | 100-1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A010670 | PGDB_C012316 | PGDB_AS002152 | View | |
| Emax | - | = | 50-120 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A036192 | PGDB_C012316 | PGDB_AS001769 | View | |
| Emax | - | < | 50 | % | - | 2 h | ALK | CRBN | - | WO2026015344A1 | PGDB_A049347 | PGDB_C012316 | PGDB_AS001094 | View | |
| EC50 | - | > | 1000 | nM | - | — | ALK | CRBN | - | WO2026015344A1 | PGDB_A076842 | PGDB_C012316 | PGDB_AS000738 | View |