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Compound
PGDB_C002285
3 activity records1 related patents
2D structure
COc1ccc2c(c1)nc([C@H]1CC[C@H](N(C)C(=O)c3cc(CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)ccn3)CC1)n2CCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 100-1000 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A015122 | PGDB_C002285 | PGDB_AS002200 | View |
| GI50 | - | = | 100-1000 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A035540 | PGDB_C002285 | PGDB_AS001555 | View |
| GI50 | - | = | 1.3 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A038318 | PGDB_C002285 | PGDB_AS000205 | View |