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SIMM · NJU
Assay
PGDB_AS002358
System: cell_based
Cell line: HEK293
Assay context summary
Assay context
82 activity records
Assay family
% Degradation
System
cell_based
Readout
Dmax
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
82 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Dmax
-
=
47.5
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A007358
PGDB_C011745
PGDB_AS002358
View
Dmax
-
=
61.9
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A007551
PGDB_C011755
PGDB_AS002358
View
Dmax
-
=
54.5
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A011066
PGDB_C011752
PGDB_AS002358
View
Dmax
-
=
51.7
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A011904
PGDB_C011761
PGDB_AS002358
View
Dmax
-
=
53.3
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A012911
PGDB_C011704
PGDB_AS002358
View
Dmax
-
=
63.4
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A015850
PGDB_C011720
PGDB_AS002358
View
Dmax
-
=
54.7
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A016473
PGDB_C011763
PGDB_AS002358
View
Dmax
-
=
59.2
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A016549
PGDB_C011722
PGDB_AS002358
View
Dmax
-
=
75.6
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A017461
PGDB_C011768
PGDB_AS002358
View
Dmax
-
=
72.8
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A018480
PGDB_C011703
PGDB_AS002358
View
Dmax
-
=
61.6
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A018947
PGDB_C011708
PGDB_AS002358
View
Dmax
-
=
55.2
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A019662
PGDB_C011762
PGDB_AS002358
View
Dmax
-
=
70.8
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A020794
PGDB_C011728
PGDB_AS002358
View
Dmax
-
=
61.9
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A021643
PGDB_C011694
PGDB_AS002358
View
Dmax
-
=
58.9
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A022294
PGDB_C011707
PGDB_AS002358
View
Dmax
-
=
51.4
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A023042
PGDB_C011766
PGDB_AS002358
View
Dmax
-
=
60.6
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A024165
PGDB_C011742
PGDB_AS002358
View
Dmax
-
=
56.4
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A024203
PGDB_C011716
PGDB_AS002358
View
Dmax
-
=
62.2
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A024249
PGDB_C011699
PGDB_AS002358
View
Dmax
-
=
39.2
%
-
24 h
CDK2
-
HEK293
WO2025224249A1
PGDB_A024407
PGDB_C011747
PGDB_AS002358
View