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Compound
PGDB_C011742
3 activity records1 related patents
2D structure
C[C@@H]1[C@@H](Nc2nnc(-c3cc(C4(C)CC4)on3)o2)CN1c1cc(F)c(C2CCC(=O)NC2=O)c(F)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 60.6 | % | - | 24 h | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A024165 | PGDB_C011742 | PGDB_AS002358 | View |
| Dmax | - | = | 14.7 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025224249A1 | PGDB_A050775 | PGDB_C011742 | PGDB_AS001257 | View |
| DC50 | - | = | 879.1 | nM | - | — | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A056526 | PGDB_C011742 | PGDB_AS000391 | View |