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Compound
PGDB_C011708
3 activity records1 related patents
2D structure
COc1c(N2C[C@H](Nc3nnc(C45CC(C(F)(F)F)(C4)C5)o3)[C@H]2C)ccc(C2CCC(=O)NC2=O)c1ClCompound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 61.6 | % | - | 24 h | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A018947 | PGDB_C011708 | PGDB_AS002358 | View |
| Dmax | - | = | 8.7 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025224249A1 | PGDB_A048894 | PGDB_C011708 | PGDB_AS001257 | View |
| DC50 | - | = | 174.1 | nM | - | — | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A076487 | PGDB_C011708 | PGDB_AS000391 | View |