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Compound
PGDB_C011752
3 activity records1 related patents
2D structure
O=C1CCC(c2c(F)cc(N3CC(Nc4nnc(C56CC(C(F)(F)F)(C5)C6)o4)C3)c(Cl)c2F)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Dmax | - | = | 54.5 | % | - | 24 h | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A011066 | PGDB_C011752 | PGDB_AS002358 | View |
| Dmax | - | = | 6.2 | % | - | 24 h | GSPT1 | - | HEK293 | WO2025224249A1 | PGDB_A040217 | PGDB_C011752 | PGDB_AS001257 | View |
| DC50 | - | = | 54.7 | nM | - | — | CDK2 | - | HEK293 | WO2025224249A1 | PGDB_A058890 | PGDB_C011752 | PGDB_AS000391 | View |