Assay
PGDB_AS002383
System: cell_basedCell line: MM.1S
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 3.3 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A009990 | PGDB_C001162 | PGDB_AS002383 | View | |
| IC50 | - | = | 17.2 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A021124 | PGDB_C001165 | PGDB_AS002383 | View | |
| IC50 | - | = | 79.6 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A025202 | PGDB_C001158 | PGDB_AS002383 | View | |
| IC50 | - | = | 29.3 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A027216 | PGDB_C001156 | PGDB_AS002383 | View | |
| IC50 | - | = | 69.9 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A033810 | PGDB_C001166 | PGDB_AS002383 | View | |
| IC50 | - | = | 98.1 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A042329 | PGDB_C001167 | PGDB_AS002383 | View | |
| IC50 | - | = | 46.9 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A051193 | PGDB_C008731 | PGDB_AS002383 | View | |
| IC50 | - | = | 39.5 | nM | - | — | - | - | MM.1S | WO2023151635A1 | PGDB_A058373 | PGDB_C001161 | PGDB_AS002383 | View |