Assay
PGDB_AS002456
System: cell_basedCell line: MV-4-11
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | <= 3 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A013490 | PGDB_C000716 | PGDB_AS002456 | View | |
| IC50 | - | = | <= 3 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A015530 | PGDB_C000725 | PGDB_AS002456 | View | |
| IC50 | - | = | > 3-5 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A021538 | PGDB_C000708 | PGDB_AS002456 | View | |
| IC50 | - | = | > 20-30 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A028240 | PGDB_C000707 | PGDB_AS002456 | View | |
| IC50 | - | = | > 3-5 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A034055 | PGDB_C000713 | PGDB_AS002456 | View | |
| IC50 | - | = | > 3-5 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A036947 | PGDB_C000714 | PGDB_AS002456 | View | |
| IC50 | - | = | > 3-5 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A058624 | PGDB_C000717 | PGDB_AS002456 | View | |
| IC50 | - | = | > 3-5 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A058867 | PGDB_C000700 | PGDB_AS002456 | View | |
| IC50 | - | = | <= 3 | nM | - | — | GSPT1 | - | MV-4-11 | CN120289428A | PGDB_A059518 | PGDB_C000058 | PGDB_AS002456 | View |