Assay context summary

Assay context

33 activity records
Activity compounds and values

Activity records

33 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000485
IC50-=8720nM-GSPT1-H1299CN117917402APGDB_A007432PGDB_C000485PGDB_AS002493View
2D structure for PGDB_C000486
IC50-=570nM-GSPT1-H1299CN117917402APGDB_A011495PGDB_C000486PGDB_AS002493View
2D structure for PGDB_C000502
IC50-=6752nM-GSPT1-H1299CN117917402APGDB_A013472PGDB_C000502PGDB_AS002493View
2D structure for PGDB_C000494
IC50-=7066nM-GSPT1-H1299CN117917402APGDB_A020024PGDB_C000494PGDB_AS002493View
2D structure for PGDB_C000490
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A020732PGDB_C000490PGDB_AS002493View
2D structure for PGDB_C000489
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A020762PGDB_C000489PGDB_AS002493View
2D structure for PGDB_C000499
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A023601PGDB_C000499PGDB_AS002493View
2D structure for PGDB_C000495
IC50-=563.7nM-GSPT1-H1299CN117917402APGDB_A024962PGDB_C000495PGDB_AS002493View
2D structure for PGDB_C000503
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A027411PGDB_C000503PGDB_AS002493View
2D structure for PGDB_C000500
IC50-=55.35nM-GSPT1-H1299CN117917402APGDB_A031148PGDB_C000500PGDB_AS002493View
2D structure for PGDB_C000476
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A031584PGDB_C000476PGDB_AS002493View
2D structure for PGDB_C000501
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A032212PGDB_C000501PGDB_AS002493View
2D structure for PGDB_C000488
IC50-=4009nM-GSPT1-H1299CN117917402APGDB_A032991PGDB_C000488PGDB_AS002493View
2D structure for PGDB_C000473
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A034012PGDB_C000473PGDB_AS002493View
2D structure for PGDB_C000477
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A036183PGDB_C000477PGDB_AS002493View
2D structure for PGDB_C000474
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A036956PGDB_C000474PGDB_AS002493View
2D structure for PGDB_C000505
IC50-=1840nM-GSPT1-H1299CN117917402APGDB_A041683PGDB_C000505PGDB_AS002493View
2D structure for PGDB_C000496
IC50-=771.1nM-GSPT1-H1299CN117917402APGDB_A044241PGDB_C000496PGDB_AS002493View
2D structure for PGDB_C000484
IC50->10000nM-GSPT1-H1299CN117917402APGDB_A047539PGDB_C000484PGDB_AS002493View
2D structure for PGDB_C000487
IC50-=2050nM-GSPT1-H1299CN117917402APGDB_A048225PGDB_C000487PGDB_AS002493View