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Cc1c(Cl)cc(NC(=O)CCc2ccc3c(c2)C(=O)N(C2CCC(=O)NC2=O)C3)cc1CN1CC2(COC2)C1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 86.4 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A009268 | PGDB_C000487 | PGDB_AS002566 | View | |
| IC50 | - | = | 55.39 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A044624 | PGDB_C000487 | PGDB_AS002565 | View | |
| IC50 | - | = | 2050 | nM | - | — | GSPT1 | - | H1299 | CN117917402A | PGDB_A048225 | PGDB_C000487 | PGDB_AS002493 | View | |
| IC50 | - | = | 31.79 | nM | - | — | - | - | MOLT-4 | CN117917402A | PGDB_A068527 | PGDB_C000487 | PGDB_AS002289 | View | |
| IC50 | - | = | 4.283 | nM | - | — | GSPT1 | - | MV-4-11 | CN117917402A | PGDB_A070025 | PGDB_C000487 | PGDB_AS000703 | View |