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COCCN(C)Cc1cc(NC(=O)CCc2cc3c(cc2F)CN(C2CCC(=O)NC2=O)C3=O)cc(Cl)c1C| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 89 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A036149 | PGDB_C000505 | PGDB_AS002565 | View | |
| IC50 | - | = | 1840 | nM | - | — | GSPT1 | - | H1299 | CN117917402A | PGDB_A041683 | PGDB_C000505 | PGDB_AS002493 | View | |
| IC50 | - | = | 97 | nM | - | — | GSPT1 | - | MV-4-11 | CN117917402A | PGDB_A045129 | PGDB_C000505 | PGDB_AS000703 | View | |
| DC50 | - | = | 21 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A046214 | PGDB_C000505 | PGDB_AS002566 | View | |
| IC50 | - | = | 18 | nM | - | — | - | - | MOLT-4 | CN117917402A | PGDB_A064822 | PGDB_C000505 | PGDB_AS002289 | View |