Assay

PGDB_AS002526

System: cell_basedTarget: KRAS
Assay context summary

Assay context

58 activity records
Assay family% Degradation
Systemcell_based
ReadoutDC50
TargetKRAS
E3Not specified
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

58 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C031991
DC50-=2.9nM-—KRAS--WO2026114958A1PGDB_A000102PGDB_C031991PGDB_AS002526View
2D structure for PGDB_C031978
DC50-=3.6nM-—KRAS--WO2026114958A1PGDB_A000531PGDB_C031978PGDB_AS002526View
2D structure for PGDB_C031966
DC50-=14.2nM-—KRAS--WO2026114958A1PGDB_A000551PGDB_C031966PGDB_AS002526View
2D structure for PGDB_C031954
DC50-=9.8nM-—KRAS--WO2026114958A1PGDB_A000593PGDB_C031954PGDB_AS002526View
2D structure for PGDB_C031946
DC50-=4.3nM-—KRAS--WO2026114958A1PGDB_A000777PGDB_C031946PGDB_AS002526View
2D structure for PGDB_C031949
DC50-=1.6nM-—KRAS--WO2026114958A1PGDB_A001148PGDB_C031949PGDB_AS002526View
2D structure for PGDB_C031961
DC50-=13.2nM-—KRAS--WO2026114958A1PGDB_A001852PGDB_C031961PGDB_AS002526View
2D structure for PGDB_C031975
DC50-=4.5nM-—KRAS--WO2026114958A1PGDB_A002102PGDB_C031975PGDB_AS002526View
2D structure for PGDB_C031960
DC50-=1.8nM-—KRAS--WO2026114958A1PGDB_A002108PGDB_C031960PGDB_AS002526View
2D structure for PGDB_C031976
DC50-=4.5nM-—KRAS--WO2026114958A1PGDB_A002473PGDB_C031976PGDB_AS002526View
2D structure for PGDB_C031983
DC50-=8.8nM-—KRAS--WO2026114958A1PGDB_A002505PGDB_C031983PGDB_AS002526View
2D structure for PGDB_C031989
DC50-=8nM-—KRAS--WO2026114958A1PGDB_A002512PGDB_C031989PGDB_AS002526View
2D structure for PGDB_C031985
DC50-=0.8nM-—KRAS--WO2026114958A1PGDB_A002541PGDB_C031985PGDB_AS002526View
2D structure for PGDB_C031992
DC50-=5.3nM-—KRAS--WO2026114958A1PGDB_A002803PGDB_C031992PGDB_AS002526View
2D structure for PGDB_C031988
DC50-=11.1nM-—KRAS--WO2026114958A1PGDB_A002984PGDB_C031988PGDB_AS002526View
2D structure for PGDB_C031943
DC50-=1.5nM-—KRAS--WO2026114958A1PGDB_A003080PGDB_C031943PGDB_AS002526View
2D structure for PGDB_C031944
DC50-=2.6nM-—KRAS--WO2026114958A1PGDB_A003174PGDB_C031944PGDB_AS002526View
2D structure for PGDB_C031955
DC50-=11.1nM-—KRAS--WO2026114958A1PGDB_A003187PGDB_C031955PGDB_AS002526View
2D structure for PGDB_C031962
DC50-=2.8nM-—KRAS--WO2026114958A1PGDB_A003697PGDB_C031962PGDB_AS002526View
2D structure for PGDB_C031950
DC50-=14.8nM-—KRAS--WO2026114958A1PGDB_A003749PGDB_C031950PGDB_AS002526View
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