Assay
PGDB_AS002551
System: cell_basedCell line: MM.1S
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A032229 | PGDB_C025807 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A034110 | PGDB_C025808 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A034568 | PGDB_C025803 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A041666 | PGDB_C015982 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A047677 | PGDB_C025815 | PGDB_AS002551 | View | |
| IC50 | - | = | 100-500 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A048831 | PGDB_C025814 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A056292 | PGDB_C025813 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A064585 | PGDB_C019593 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A066129 | PGDB_C025806 | PGDB_AS002551 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MM.1S | CN116239566A | PGDB_A068518 | PGDB_C025809 | PGDB_AS002551 | View |