PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Assay
PGDB_AS002552
System: cell_based
Target: CRBN
Assay context summary
Assay context
406 activity records
Assay family
biochemical
System
cell_based
Readout
% Inhibition
Target
CRBN
E3
CRBN
Organism
Homo sapiens
Technology
HTRF
Detection target
cell_inhibition
Activity compounds and values
Activity records
406 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081916
PGDB_C022139
PGDB_AS002552
View
% Inhibition
-
=
53-60
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081938
PGDB_C021982
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081949
PGDB_C022327
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081974
PGDB_C022046
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081975
PGDB_C022087
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081984
PGDB_C022112
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A081985
PGDB_C022109
PGDB_AS002552
View
% Inhibition
-
=
53-60
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082004
PGDB_C022331
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082014
PGDB_C022039
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082015
PGDB_C022410
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082031
PGDB_C022418
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082048
PGDB_C022305
PGDB_AS002552
View
% Inhibition
-
=
53-60
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082052
PGDB_C022132
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082075
PGDB_C022348
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082081
PGDB_C022272
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082086
PGDB_C022296
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082087
PGDB_C022004
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082091
PGDB_C022230
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082092
PGDB_C022324
PGDB_AS002552
View
% Inhibition
-
=
60-80
%
2 uM
3 h
CRBN
CRBN
-
CN119654316A
PGDB_A082094
PGDB_C022390
PGDB_AS002552
View