Assay context summary

Assay context

33 activity records
Activity compounds and values

Activity records

33 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000501
IC50->10000nM-GSPT1-U937CN117917402APGDB_A008444PGDB_C000501PGDB_AS002565View
2D structure for PGDB_C000494
IC50-=291.9nM-GSPT1-U937CN117917402APGDB_A010847PGDB_C000494PGDB_AS002565View
2D structure for PGDB_C000474
IC50-=31.37nM-GSPT1-U937CN117917402APGDB_A015083PGDB_C000474PGDB_AS002565View
2D structure for PGDB_C000496
IC50-=27.2nM-GSPT1-U937CN117917402APGDB_A015483PGDB_C000496PGDB_AS002565View
2D structure for PGDB_C000482
IC50-=3301nM-GSPT1-U937CN117917402APGDB_A016071PGDB_C000482PGDB_AS002565View
2D structure for PGDB_C000488
IC50-=106.1nM-GSPT1-U937CN117917402APGDB_A018645PGDB_C000488PGDB_AS002565View
2D structure for PGDB_C000477
IC50-=321nM-GSPT1-U937CN117917402APGDB_A023308PGDB_C000477PGDB_AS002565View
2D structure for PGDB_C000485
IC50-=81.79nM-GSPT1-U937CN117917402APGDB_A024314PGDB_C000485PGDB_AS002565View
2D structure for PGDB_C000489
IC50-=81.52nM-GSPT1-U937CN117917402APGDB_A026144PGDB_C000489PGDB_AS002565View
2D structure for PGDB_C000492
IC50-=87.18nM-GSPT1-U937CN117917402APGDB_A026479PGDB_C000492PGDB_AS002565View
2D structure for PGDB_C000473
IC50-=179.5nM-GSPT1-U937CN117917402APGDB_A033195PGDB_C000473PGDB_AS002565View
2D structure for PGDB_C000500
IC50-=11.2nM-GSPT1-U937CN117917402APGDB_A035075PGDB_C000500PGDB_AS002565View
2D structure for PGDB_C000486
IC50-=11nM-GSPT1-U937CN117917402APGDB_A035912PGDB_C000486PGDB_AS002565View
2D structure for PGDB_C000505
IC50-=89nM-GSPT1-U937CN117917402APGDB_A036149PGDB_C000505PGDB_AS002565View
2D structure for PGDB_C000481
IC50->10000nM-GSPT1-U937CN117917402APGDB_A037863PGDB_C000481PGDB_AS002565View
2D structure for PGDB_C000484
IC50-=401.7nM-GSPT1-U937CN117917402APGDB_A040282PGDB_C000484PGDB_AS002565View
2D structure for PGDB_C000498
IC50-=905.4nM-GSPT1-U937CN117917402APGDB_A040690PGDB_C000498PGDB_AS002565View
2D structure for PGDB_C000493
IC50-=141nM-GSPT1-U937CN117917402APGDB_A042156PGDB_C000493PGDB_AS002565View
2D structure for PGDB_C000483
IC50->10000nM-GSPT1-U937CN117917402APGDB_A043517PGDB_C000483PGDB_AS002565View
2D structure for PGDB_C000478
IC50-=1253nM-GSPT1-U937CN117917402APGDB_A044217PGDB_C000478PGDB_AS002565View