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O=C1CCC(N2Cc3ccc(CCC(=O)Nc4ccc(-c5cccnc5)c(CN5CCOCC5)c4)cc3C2=O)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 212.4 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A016636 | PGDB_C000493 | PGDB_AS002566 | View | |
| IC50 | - | = | 141 | nM | - | — | GSPT1 | - | U937 | CN117917402A | PGDB_A042156 | PGDB_C000493 | PGDB_AS002565 | View | |
| IC50 | - | = | 8.359 | nM | - | — | GSPT1 | - | MV-4-11 | CN117917402A | PGDB_A045628 | PGDB_C000493 | PGDB_AS000703 | View | |
| IC50 | - | = | 75.12 | nM | - | — | - | - | MOLT-4 | CN117917402A | PGDB_A060539 | PGDB_C000493 | PGDB_AS002289 | View | |
| IC50 | - | > | 10000 | nM | - | — | GSPT1 | - | H1299 | CN117917402A | PGDB_A068316 | PGDB_C000493 | PGDB_AS002493 | View |