Summary
AssigneeCelgene
Filing years2019-2020
Patents2
Compounds9
Activity records38
Patent families2
Targets5
Assay familiesbinding, degradation
Activity metricsIC50, inhibition
Overview

Target distribution and active-compound trend

Target distribution

41 activity records

6 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

03620202024
Activity compounds and values

Activity records

41 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C005650
IC50-=0.08nM-IKZF3CRBNOPM-2AU2019272751B2PGDB_A007476PGDB_C005650PGDB_AS002253View
2D structure for PGDB_C005650
IC50-=0.13nM-IKZF1CRBNOPM-2AU2019272751B2PGDB_A008496PGDB_C005650PGDB_AS000106View
2D structure for PGDB_C019024
IC50->100nM-IKZF1CRBNOPM-2AU2019272751B2PGDB_A009428PGDB_C019024PGDB_AS000106View
2D structure for PGDB_C019024
IC50->100nM-IKZF1CRBNOPM-2AU2019272751B2PGDB_A010160PGDB_C019024PGDB_AS001658View
2D structure for PGDB_C019024
IC50->100nM-ZFP91CRBNOPM-2AU2019272751B2PGDB_A012772PGDB_C019024PGDB_AS000285View
2D structure for PGDB_C009601
IC50-=89nM-IKZF3CRBNOPM-2AU2019272751B2PGDB_A012964PGDB_C009601PGDB_AS002253View
2D structure for PGDB_C005650
IC50-=0.06nM-IKZF3-OPM-2AU2019272751B2PGDB_A019381PGDB_C005650PGDB_AS001698View
2D structure for PGDB_C005650
IC50-=0.08nM-ZFP91CRBNOPM-2AU2019272751B2PGDB_A021546PGDB_C005650PGDB_AS000285View
2D structure for PGDB_C005651
IC50-=0.0059uM-IKZF3CRBNDF15AU2019272751B2PGDB_A023925PGDB_C005651PGDB_AS001348View
2D structure for PGDB_C005651
IC50->0.1uM-IKZF3CRBNDF15AU2019272751B2PGDB_A026335PGDB_C005651PGDB_AS001313View
2D structure for PGDB_C005650
IC50->100nM-IKZF1CRBNOPM-2AU2019272751B2PGDB_A030612PGDB_C005650PGDB_AS001658View
2D structure for PGDB_C009601
IC50-=91nM-IKZF1CRBNOPM-2AU2019272751B2PGDB_A031052PGDB_C009601PGDB_AS000106View
2D structure for PGDB_C009601
IC50-=56nM-IKZF3-OPM-2AU2019272751B2PGDB_A035209PGDB_C009601PGDB_AS001698View
2D structure for PGDB_C009601
IC50->100nM-IKZF1CRBNOPM-2AU2019272751B2PGDB_A039396PGDB_C009601PGDB_AS001658View
2D structure for PGDB_C019024
IC50->100nM-IKZF3-OPM-2AU2019272751B2PGDB_A040345PGDB_C019024PGDB_AS001698View
2D structure for PGDB_C009601
IC50->100nM-IKZF1-OPM-2AU2019272751B2PGDB_A040978PGDB_C009601PGDB_AS000771View
2D structure for PGDB_C005650
IC50-=0.08nM--CRBNOPM-2AU2019272751B2PGDB_A044255PGDB_C005650PGDB_AS002367View
2D structure for PGDB_C005650
IC50->0.1uM-IKZF3CRBNDF15AU2019272751B2PGDB_A044432PGDB_C005650PGDB_AS001313View
2D structure for PGDB_C005651
IC50-=0.00045uM-IKZF3CRBNDF15AU2019272751B2PGDB_A048390PGDB_C005651PGDB_AS002160View
2D structure for PGDB_C005650
IC50-=0.000031uM-IKZF3CRBNDF15AU2019272751B2PGDB_A049649PGDB_C005650PGDB_AS002160View