Summary
AssigneeChina Pharmaceutical University
Filing years2023-2025
Patents7
Compounds211
Activity records512
Patent families7
Targets5
Assay familiesbinding, cellular_function, degradation, viability
Activity metricsDC50, IC50, Ki, degradation, inhibition
Overview

Target distribution and active-compound trend

Target distribution

512 activity records

5 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

04895202420252026
Activity compounds and values

Activity records

512 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C006929
% Degradation-=39%--VHL-SH-SY5YCN119613482APGDB_A011154PGDB_C006929PGDB_AS001892View
2D structure for PGDB_C006936
Ki-<300nM-VHLVHL-CN119613482APGDB_A011709PGDB_C006936PGDB_AS000103View
2D structure for PGDB_C006937
% Degradation-=28%--VHL-SH-SY5YCN119613482APGDB_A012032PGDB_C006937PGDB_AS001892View
2D structure for PGDB_C006933
% Degradation-=40%--VHL-SH-SY5YCN119613482APGDB_A021761PGDB_C006933PGDB_AS001892View
2D structure for PGDB_C006925
% Degradation-=80%--VHL-SH-SY5YCN119613482APGDB_A022677PGDB_C006925PGDB_AS001892View
2D structure for PGDB_C006934
Ki-<300nM-VHLVHL-CN119613482APGDB_A023786PGDB_C006934PGDB_AS000103View
2D structure for PGDB_C006928
% Degradation-=82%--VHL-SH-SY5YCN119613482APGDB_A024284PGDB_C006928PGDB_AS001892View
2D structure for PGDB_C006928
Ki-<300nM-VHLVHL-CN119613482APGDB_A029167PGDB_C006928PGDB_AS000103View
2D structure for PGDB_C006934
% Degradation-=54%--VHL-SH-SY5YCN119613482APGDB_A030754PGDB_C006934PGDB_AS001892View
2D structure for PGDB_C006937
Ki-<300nM-VHLVHL-CN119613482APGDB_A035537PGDB_C006937PGDB_AS000103View
2D structure for PGDB_C006931
Ki-<300nM-VHLVHL-CN119613482APGDB_A035851PGDB_C006931PGDB_AS000103View
2D structure for PGDB_C006931
% Degradation-=56%--VHL-SH-SY5YCN119613482APGDB_A036890PGDB_C006931PGDB_AS001892View
2D structure for PGDB_C006930
Ki-<300nM-VHLVHL-CN119613482APGDB_A038856PGDB_C006930PGDB_AS000103View
2D structure for PGDB_C006924
Ki-<300nM-VHLVHL-CN119613482APGDB_A041491PGDB_C006924PGDB_AS000103View
2D structure for PGDB_C006935
Ki-<300nM-VHLVHL-CN119613482APGDB_A044712PGDB_C006935PGDB_AS000103View
2D structure for PGDB_C006935
% Degradation-=32%--VHL-SH-SY5YCN119613482APGDB_A045639PGDB_C006935PGDB_AS001892View
2D structure for PGDB_C006932
Ki-<300nM-VHLVHL-CN119613482APGDB_A046111PGDB_C006932PGDB_AS000103View
2D structure for PGDB_C006924
% Degradation-=68%--VHL-SH-SY5YCN119613482APGDB_A047248PGDB_C006924PGDB_AS001892View
2D structure for PGDB_C006933
Ki-<300nM-VHLVHL-CN119613482APGDB_A051045PGDB_C006933PGDB_AS000103View
2D structure for PGDB_C006932
% Degradation-=32%--VHL-SH-SY5YCN119613482APGDB_A052437PGDB_C006932PGDB_AS001892View