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Compound
PGDB_C000356
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3cc(CNC(=O)c4ccc(C(=O)c5ccccc5)cc4)ccc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 67.3 | nM | - | — | - | - | Raji | CN117683022A | PGDB_A026802 | PGDB_C000356 | PGDB_AS000751 | View |
| IC50 | - | = | 123.1 | nM | - | — | - | - | THP-1 | CN117683022A | PGDB_A029250 | PGDB_C000356 | PGDB_AS000289 | View |
| % Degradation | - | = | 60-80 | % | 1 uM | - | GSPT1 | - | - | CN117683022A | PGDB_A041441 | PGDB_C000356 | PGDB_AS001783 | View |
| % Degradation | - | = | 30-60 | % | 1 uM | - | BRD4 | - | - | CN117683022A | PGDB_A077553 | PGDB_C000356 | PGDB_AS002272 | View |