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Compound
PGDB_C002208
4 activity records1 related patents
2D structure
Cn1c(C2CCC(NC(=O)C3CC(CNc4cccc5c4C(=O)N(C4CCC(=O)NC4=O)C5=O)C3)CC2)nc2ccncc21Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 19.61 | nM | - | — | GSPT1 | - | Toledo | WO2023237116A1 | PGDB_A014474 | PGDB_C002208 | PGDB_AS002036 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A046150 | PGDB_C002208 | PGDB_AS002200 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A048139 | PGDB_C002208 | PGDB_AS001555 | View |
| GI50 | - | = | 6.91 | nM | - | — | GSPT1 | - | NCI-H929 | WO2023237116A1 | PGDB_A064180 | PGDB_C002208 | PGDB_AS000710 | View |