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Compound
PGDB_C002254
5 activity records1 related patents
2D structure
Cn1c2cnccc2nc1[C@H]1CC[C@H](NC(=O)c2cc(CNc3cccc4c3C(=O)N(C3CCC(=O)NC3=O)C4=O)ccn2)CC1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 3.58 | nM | - | — | GSPT1 | - | Raji | WO2023237116A1 | PGDB_A015810 | PGDB_C002254 | PGDB_AS000230 | View |
| GI50 | - | = | 1.73 | nM | - | — | GSPT1 | - | SU-DHL-2 | WO2023237116A1 | PGDB_A057236 | PGDB_C002254 | PGDB_AS000205 | View |
| DC50 | - | < | 100 | nM | - | — | GSPT1 | - | HEK293 | WO2023237116A1 | PGDB_A067451 | PGDB_C002254 | PGDB_AS002200 | View |
| GI50 | - | = | 0.99 | nM | - | — | GSPT1 | - | NCI-H929 | WO2023237116A1 | PGDB_A069795 | PGDB_C002254 | PGDB_AS000710 | View |
| GI50 | - | < | 100 | nM | - | — | GSPT1 | - | HL-60 | WO2023237116A1 | PGDB_A073620 | PGDB_C002254 | PGDB_AS001555 | View |